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Cobimetinib R-enantiomer
CAS No. 934660-94-3
Cobimetinib R-enantiomer( GDC-0973 R-enantiomer | XL-518 R-enantiomer )
Catalog No. M16683 CAS No. 934660-94-3
Cobimetinib R-enantiomer (GDC-0973; XL518) is the R-enantiomer of Cobimetinib (GDC-0973; XL518).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 1153 | Get Quote |
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| 100MG | Get Quote | Get Quote |
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| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameCobimetinib R-enantiomer
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NoteResearch use only, not for human use.
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Brief DescriptionCobimetinib R-enantiomer (GDC-0973; XL518) is the R-enantiomer of Cobimetinib (GDC-0973; XL518).
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DescriptionCobimetinib R-enantiomer (GDC-0973; XL518) is the R-enantiomer of Cobimetinib (GDC-0973; XL518), which is a potent, highly selective inhibitor of mitogen-activated protein kinase kinase(MEK1/2).
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In Vitro——
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In Vivo——
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SynonymsGDC-0973 R-enantiomer | XL-518 R-enantiomer
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PathwayMAPK/ERK Signaling
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TargetMEK
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RecptorMEK
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number934660-94-3
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Formula Weight531.31
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Molecular FormulaC21H21F3IN3O2
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Purity>98% (HPLC)
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Solubility10 mM in DMSO
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SMILESFC1=C(F)C=CC(C(N2CC([C@H]3CCCCN3)(O)C2)=O)=C1NC4=CC=C(I)C=C4F
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Chemical NameMethanone, [3,4-difluoro-2-[(2-fluoro-4-iodophenyl)amino]phenyl][3-hydroxy-3-[(2R)-2-piperidinyl]-1-azetidinyl]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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